SCHEMBL2310282

SCHEMBL2310282

Cc1cc(Cn2c(C)c(C(=O)O)c3c([C@@H](c4cccc(F)c4C(N)=O)C4CC4)ccc(F)c3c2=O)no1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.38
TRPA1 O75762 5/20 0.34
S1PR3 Q99500 2/20 0.34
GRIN1 Q05586 4/20 0.32
GRIN2B Q13224 4/20 0.32
GLP1R P43220 1/20 0.32
REN P00797 1/20 0.32
KCNH2 Q12809 1/20 0.32
GABRA5 P31644 2/20 0.32
GABRA1 P14867 1/20 0.32
DPP4 P27487 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE1C Q14123 1/20 0.31
MAPT P10636 1/20 0.31
RECQL P46063 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2311690 0.87 GNRHR (0.35)
SCHEMBL2356247 0.85 MAPT (0.31) GRIN1GRIN2BDPP4MAPT
SCHEMBL2308354 0.84 S1PR3 (0.33) S1PR3GLP1RRENKCNH2
SCHEMBL2313425 0.83 GNRHR (0.39) FEN1S1PR3GRIN1GRIN2B
SCHEMBL2313391 0.81 S1PR3 (0.34) S1PR3GLP1R
SCHEMBL2309555 0.76 FEN1 (0.48) FEN1TRPA1S1PR3GRIN1GRIN2B
SCHEMBL2310390 0.76 CYP2C9 (0.39)
SCHEMBL3380867 0.74 CYP2C9 (0.36) GRIN1GRIN2B
SCHEMBL2306989 0.74 S1PR3 (0.35) S1PR3GLP1R
SCHEMBL2312871 0.73 CYP2C9 (0.39) S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350015-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2011-08-03 EP claimed