SCHEMBL23075419

SCHEMBL23075419

CC(C)(C)OC(=O)n1cc(Cc2cccc(F)n2)cn1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 15/20 0.45
SCD O00767 1/20 0.38
MGLL Q99685 1/20 0.38
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29842599 1.00 RIPK1 (0.45) RIPK1SCDMGLLROCK2
SCHEMBL23075373 0.87 RIPK1 (0.43) RIPK1SCDMGLLROCK2
SCHEMBL29842646 0.87 RIPK1 (0.43) RIPK1SCDMGLLROCK2
SCHEMBL29842703 0.86 RIPK1 (0.47) RIPK1SCDMGLLROCK2
SCHEMBL23085661 0.86 RIPK1 (0.47) RIPK1SCDMGLLROCK2
SCHEMBL23067796 0.82 RIPK1 (0.46) RIPK1
SCHEMBL29842483 0.81 RIPK1 (0.42) RIPK1SCDMGLLROCK2
SCHEMBL23075410 0.81 RIPK1 (0.42) RIPK1SCDMGLLROCK2
SCHEMBL23075460 0.80 RIPK1 (0.43) RIPK1SCDMGLLROCK2
SCHEMBL28707994 0.80 GPR119 (0.42) RIPK1SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117083270-A Heterocyclic RIP1 kinase inhibitors 里格尔药品股份有限公司 2023-11-17 CN disclosed
US-20230057341-A1 HETEROCYCLIC RIP1 KINASE INHIBITORS RIGEL PHARMACEUTICALS, INC. 2023-02-23 US disclosed
CN-114761398-A Heterocyclic RIP1 kinase inhibitors 里格尔药品股份有限公司 2022-07-15 CN disclosed
US-20210070744-A1 HETEROCYCLIC RIP1 KINASE INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2021-03-11 US disclosed
WO-2021046447-A1 HETEROCYCLIC RIP1 KINASE INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2021-03-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210070744-A1 HETEROCYCLIC RIP1 KINASE INHIBITORS RIPK1, RIPK2, RIPK3 RIPK1 1/4885SCD 1636/4885MGLL 3330/4885
US-20230057341-A1 HETEROCYCLIC RIP1 KINASE INHIBITORS RIPK1, RIPK2, RIPK3 RIPK1 1/4885SCD 1636/4885MGLL 3330/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.