SCHEMBL2307993

SCHEMBL2307993

[CH2]CCC1CCCCN1S(=O)(=O)c1c(C)cc(OC)cc1C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
PSEN1 P49768 2/20 0.41
PSEN2 P49810 2/20 0.41
APH1B Q8WW43 2/20 0.41
NCSTN Q92542 2/20 0.41
APH1A Q96BI3 2/20 0.41
PSENEN Q9NZ42 2/20 0.41
CASP1 P29466 1/20 0.39
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
BDKRB1 P46663 1/20 0.38
FKBP1A P62942 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13649888 0.89 PSEN1 (0.53) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL10246104 0.88 NPC1 (0.43) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL4404580 0.87 PSEN1 (0.46) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL2934286 0.86 HTR7 (0.40) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL639859 0.86 NPC1 (0.42) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL639468 0.86 HTR7 (0.41) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL3313366 0.85 CNR2 (0.43) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL640463 0.85 RAB9A (0.41) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL639832 0.85 CNR2 (0.43) HTR7TMEM97SIGMAR1NPC1RAB9A
SCHEMBL13368948 0.85 HTR7 (0.41) HTR7TMEM97SIGMAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350003-A1 SUBSTITUTED DISULFONAMIDES AS BRI-MODULATORS Grünenthal GmbH (DE) 2011-08-03 EP disclosed
WO-2010051977-A1 SUBSTITUTED DISULFONAMIDES AS BRI-MODULATORS Grünenthal GmbH (DE) 2010-05-14 WO disclosed