Bicarbonate

Bicarbonate

SCHEMBL2308696

O=C(O)O.O=C(c1ccc(-c2ccc(Nc3nc4ccc(F)cc4o3)cc2)cc1)C1CCCC1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.45
CTSS P25774 3/20 0.45
HCRTR1 O43613 4/20 0.42
CSF1R P07333 1/20 0.42
DGAT1 O75907 2/20 0.40
HDAC6 Q9UBN7 4/20 0.40
CHEK2 O96017 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
GABRA4 P48169 1/20 0.39
GABRE P78334 1/20 0.39
GABRA6 Q16445 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL2309400 0.92 HDAC6 (0.47) CTSLCTSSHCRTR1CSF1RDGAT1
Bicarbonate SCHEMBL2314871 0.89 DGAT1 (0.51) CTSLCTSSHCRTR1CSF1RDGAT1
Bicarbonate SCHEMBL2312892 0.88 HDAC6 (0.47) CSF1RDGAT1HDAC6CHEK2GABRP
Bicarbonate SCHEMBL2309024 0.88 RAB9A (0.43) CTSLCTSSCSF1RDGAT1HDAC6
Bicarbonate SCHEMBL2311872 0.87 HDAC6 (0.47) CSF1RDGAT1HDAC6CHEK2GABRP
SCHEMBL2309763 0.86 DGAT1 (0.54) CTSLCTSSHCRTR1DGAT1
SCHEMBL13760251 0.86 DGAT1 (0.54) CTSLCTSSHCRTR1DGAT1
SCHEMBL2308693 0.86 DGAT1 (0.54) CTSLCTSSHCRTR1DGAT1
SCHEMBL2310956 0.86 DGAT1 (0.54) CTSLCTSSHCRTR1DGAT1
Bicarbonate SCHEMBL2310716 0.85 NPC1 (0.53) CSF1RDGAT1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP claimed