SCHEMBL23097685

SCHEMBL23097685

Cc1ccc(N2CCN(CCCOc3ccc4[nH]c(=O)oc4c3)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.57
DRD2 P14416 6/20 0.56
DRD3 P35462 4/20 0.56
HTR1A P08908 1/20 0.56
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23097701 0.90 KCNH2 (0.70) KCNH2DRD2DRD3HTR1A
SCHEMBL2021505 0.82 KCNH2 (0.83) KCNH2KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL2021501 0.82 KCNH2 (0.83) KCNH2KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL2021499 0.82 KCNH2 (0.83) KCNH2KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL10745044 0.81 DRD2 (0.80) DRD2DRD3HTR1AKDM4EALDH1A1
SCHEMBL23097784 0.80 DRD2 (0.61) KCNH2DRD2DRD3
SCHEMBL10518689 0.78 SIGMAR1 (0.62) DRD2DRD3HTR1A
SCHEMBL23097637 0.75 DRD2 (0.58) KCNH2DRD2DRD3HTR1A
SCHEMBL19048005 0.75 KDM1A (0.63) KCNH2DRD2
SCHEMBL20372647 0.75 HRH3 (0.71) KCNH2DRD2DRD3HTR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170334-B1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION UNIV EMORY (US) 2021-03-17 EP disclosed