SCHEMBL23099404

SCHEMBL23099404

CCc1nc2ccc(C#N)cn2c1C(=O)OCC[Si](C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
PDE5A O76074 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CYP2C9 P11712 4/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 3/20 0.35
CYP1A2 P05177 1/20 0.35
ALDH1A1 P00352 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CSF1R P07333 1/20 0.34
MAPK1 P28482 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
ELANE P08246 2/20 0.32
METTL3 Q86U44 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23099653 0.88 KDM4E (0.49) KDM4EPDE5ANPC1RAB9ACYP2C9
SCHEMBL18629888 0.76 SLC22A12 (0.37) KDM4EPDE5ACYP2C9CYP3A4CYP2C19
SCHEMBL22279584 0.71 RAB9A (0.65) KDM4ENPC1RAB9ACYP2C9CYP2C19
SCHEMBL23099627 0.69 NPC1 (0.50) KDM4ENPC1RAB9ACYP2C9CYP2C19
SCHEMBL12295206 0.69 CYP2C9 (0.67) KDM4ENPC1RAB9ACYP2C9CYP3A4
SCHEMBL23099502 0.69 KDM4E (0.49) KDM4ENPC1RAB9ACYP2C9CYP2C19
SCHEMBL23197396 0.69 RAB9A (0.49) KDM4ENPC1RAB9ACYP2C9CYP2C19
SCHEMBL12294581 0.68 CYP2C9 (0.67) RAB9ACYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL23099634 0.67 RAB9A (0.47) KDM4ENPC1RAB9ACYP2C9CYP3A4
SCHEMBL12295661 0.66 CYP2C9 (0.64) CYP2C9CYP3A4CYP2C19CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021048342-A1 ANTIBACTERIAL COMPOUNDS Janssen Sciences Ireland Unlimited Company (IE) 2021-03-18 WO disclosed