SCHEMBL2310150

SCHEMBL2310150

C[CH]c1cc(N)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
NR2E1 Q9Y466 1/20 0.39
KIF11 P52732 2/20 0.34
RPS6KA3 P51812 1/20 0.34
JAK3 P52333 1/20 0.34
NFE2L2 Q16236 1/20 0.33
IDO1 P14902 3/20 0.33
TDO2 P48775 1/20 0.33
PTPN5 P54829 2/20 0.32
IKBKB O14920 1/20 0.32
ALDH1A1 P00352 2/20 0.31
MAPT P10636 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1547520 0.84 CES2 (0.41) RPS6KA3JAK3NFE2L2IDO1TDO2
SCHEMBL27585754 0.79 TSHR (0.42) TSHRMAPK1NR2E1KIF11RPS6KA3
SCHEMBL22572970 0.79 TSHR (0.42) TSHRMAPK1NR2E1KIF11RPS6KA3
SCHEMBL394717 0.77 TSHR (0.56) TSHRMAPK1NR2E1KIF11IDO1
SCHEMBL130383 0.77 TSHR (0.56) TSHRMAPK1NR2E1KIF11IDO1
Hydrochloric Acid SCHEMBL9741395 0.74 TSHR (0.54) TSHRMAPK1NR2E1KIF11IDO1
Iodide SCHEMBL31550893 0.74 TSHR (0.54) TSHRMAPK1NR2E1KIF11IDO1
SCHEMBL27859051 0.74 TSHR (0.54) TSHRMAPK1NR2E1KIF11IDO1
SCHEMBL20569493 0.72 RPS6KA3 (0.40) TSHRMAPK1NR2E1RPS6KA3JAK3
SCHEMBL3981283 0.71 CYP19A1 (0.33) TSHRNFE2L2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2348860-A1 PYRAZOLOPYRIMIDINE JAK INHIBITOR COMPOUNDS AND METHODS Genentech, Inc. (US) 2011-08-03 EP disclosed