SCHEMBL23102431

SCHEMBL23102431

Cc1c(Br)cccc1-c1nc2c(O)nccc2s1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
TP53 P04637 4/20 0.33
MAPT P10636 3/20 0.33
APP P05067 1/20 0.33
ALDH1A1 P00352 4/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
RXFP1 Q9HBX9 2/20 0.32
APOBEC3A P31941 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102434 0.73 KDM4E (0.41) KDM4ETP53MAPTALDH1A1NPC1
SCHEMBL31354064 0.73 KDM4E (0.41) KDM4ETP53MAPTALDH1A1NPC1
SCHEMBL23102399 0.73 PARP1 (0.37) KDM4EPDCD1CD274TP53MAPT
SCHEMBL23102415 0.69 PDCD1 (0.37) KDM4EPDCD1CD274TP53MAPT
SCHEMBL20477485 0.69 MAPT (0.44) KDM4EMAPTAPPALDH1A1NPC1
SCHEMBL23624312 0.67 KDM4E (0.35) KDM4EPDCD1CD274TP53MAPT
SCHEMBL24660285 0.65 LMNA (0.39) KDM4EPDCD1CD274TP53MAPT
SCHEMBL20539398 0.64 KDM4E (0.41) KDM4ETP53MAPTAPPALDH1A1
SCHEMBL20539648 0.64 HSD17B13 (0.42) PDCD1CD274S1PR1
SCHEMBL27989971 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed