SCHEMBL23624312

SCHEMBL23624312

Cc1sc(-c2cccc(Br)c2C)nc1CO

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
PDCD1 Q15116 3/20 0.35
CD274 Q9NZQ7 3/20 0.35
HTR2B P41595 1/20 0.35
TP53 P04637 3/20 0.33
MAPT P10636 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
S1PR1 P21453 1/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 4/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
AHR P35869 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469388 0.77 HTR2B (0.57) KDM4EHTR2BMAPTALDH1A1SMN1; SMN2
SCHEMBL23624231 0.75 NPC1 (0.41) KDM4EPDCD1CD274HTR2BTP53
SCHEMBL24660285 0.74 LMNA (0.39) KDM4EPDCD1CD274TP53MAPT
SCHEMBL20539648 0.73 HSD17B13 (0.42) PDCD1CD274S1PR1
SCHEMBL4034919 0.71 RARA (0.49) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL30522700 0.71 PDCD1 (0.35) KDM4EPDCD1CD274
SCHEMBL28486432 0.71 PDCD1 (0.35) KDM4EPDCD1CD274
SCHEMBL12875931 0.70 ALDH1A1 (0.46) MAPTALDH1A1MEN1RAB9AKMT2A
SCHEMBL18003926 0.69 ALDH1A1 (0.34) KDM4EPDCD1CD274MAPTALDH1A1
SCHEMBL23102434 0.69 KDM4E (0.41) KDM4ETP53MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021136354-A1 BIPHENYL DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2021-07-08 WO disclosed