SCHEMBL23102444

SCHEMBL23102444

COc1nccc2c1nc(-c1cccc(Br)c1C)n2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 2/20 0.38
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SHMT2 P34897 1/20 0.33
PARP1 P09874 1/20 0.33
CARM1 Q86X55 1/20 0.33
JAK2 O60674 2/20 0.32
TYK2 P29597 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP1A2 P05177 1/20 0.32
S1PR1 P21453 1/20 0.32
MMP12 P39900 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102443 0.71 KDM4E (0.43) PARP1JAK2KMT2ACYP1A2BTK
SCHEMBL23102647 0.66 RPS6KA5 (0.38) RPS6KA5PDE1APDE1BPDE1C
SCHEMBL18686677 0.66 SMN1; SMN2 (0.37) SMN1; SMN2CYP2C19CYP1A2
SCHEMBL20086199 0.66 ALDH1A1 (0.39) POLBSMN1; SMN2JAK2TYK2MEN1
SCHEMBL31343149 0.65 ALDH1A1 (0.44) POLBSMN1; SMN2MEN1KMT2AHSD11B1
SCHEMBL19766304 0.65 ALDH1A1 (0.44) POLBSMN1; SMN2MEN1KMT2AHSD11B1
SCHEMBL6366681 0.65 TLR8 (0.40) PARP1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL23102648 0.63 RPS6KA5 (0.44) RPS6KA5POLBCYP1A2
SCHEMBL23103161 0.63 CD274 (0.42) PDCD1CD274
SCHEMBL31004236 0.63 CD274 (0.42) PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed