SCHEMBL23102443

SCHEMBL23102443

Cc1c(Br)cccc1-c1nc2c(=O)[nH]ccc2n1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
CYP1A2 P05177 1/20 0.43
HPGD P15428 1/20 0.43
PARP1 P09874 1/20 0.37
PTGES O14684 1/20 0.35
GAA P10253 1/20 0.33
BRD1 O95696 1/20 0.32
TAF1 P21675 1/20 0.32
BRPF1 P55201 1/20 0.32
KMT2A Q03164 1/20 0.31
HSD11B1 P28845 1/20 0.31
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
JAK2 O60674 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29246381 0.74 CSNK2A2 (0.35) KDM4EALDH1A1CYP1A2HPGDPARP1
SCHEMBL23102399 0.72 PARP1 (0.37) KDM4EALDH1A1PARP1MAPT
SCHEMBL23102409 0.72 C1R (0.40) KDM4EALDH1A1HPGDPARP1KMT2A
SCHEMBL23102444 0.71 RPS6KA5 (0.38) CYP1A2PARP1KMT2AHSD11B1JAK2
SCHEMBL19766304 0.66 ALDH1A1 (0.44) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL31343149 0.66 ALDH1A1 (0.44) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL146880 0.66 KDM4E (0.37) KDM4EALDH1A1CYP1A2HPGDPARP1
SCHEMBL6366681 0.65 TLR8 (0.40) CYP1A2PARP1KMT2A
SCHEMBL23639740 0.65 CYP1A2 (0.41) KDM4EALDH1A1CYP1A2HPGDPARP1
SCHEMBL15059285 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed