SCHEMBL2310592

SCHEMBL2310592

CN(C)C(c1ccccc1)C1CCC(NS(=O)(=O)c2ccc(C(C)(C)C)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
PSEN1 P49768 1/20 0.42
PSEN2 P49810 1/20 0.42
SPPL2A Q8TCT8 1/20 0.42
APH1B Q8WW43 1/20 0.42
NCSTN Q92542 1/20 0.42
APH1A Q96BI3 1/20 0.42
PSENEN Q9NZ42 1/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
DRD3 P35462 1/20 0.42
GAA P10253 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PARG Q86W56 1/20 0.41
ALDH1A1 P00352 4/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1326592 0.99 KMT2A (0.46) KMT2APSEN1PSEN2SPPL2AAPH1B
SCHEMBL2312046 0.89 PARG (0.45) KMT2ADRD2PARGALDH1A1KDM4E
Hydrochloric Acid SCHEMBL1326995 0.88 PARG (0.44) KMT2ADRD2PARGALDH1A1KDM4E
SCHEMBL2306896 0.86 HTT (0.51) KMT2APSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL1326839 0.85 HTT (0.50) KMT2APSEN1PSEN2APH1BNCSTN
SCHEMBL2308706 0.84 MMP2 (0.48) KMT2AGAAPARGALDH1A1MEN1
Hydrochloric Acid SCHEMBL1327141 0.83 MMP2 (0.47) KMT2AGAAPARGALDH1A1MEN1
SCHEMBL9906394 0.80 KMT2A (0.66) KMT2ATDP1ALDH1A1KDM4ERECQL
SCHEMBL2356839 0.79 ALDH1A1 (0.58) KMT2ADRD2HTR2APARGALDH1A1
SCHEMBL1327484 0.78 MEN1 (0.55) KMT2ADRD2HTR2ADRD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989174-B1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES GRUENENTHAL GMBH (DE) 2011-08-03 EP claimed
JP-2009520720-A 2009-05-28 JP claimed
EP-1989174-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2008-11-12 EP claimed
WO-2007079930-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO claimed
EP-1989174-B1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES GRUENENTHAL GMBH (DE) 2011-08-03 EP disclosed
EP-1989174-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2008-11-12 EP disclosed
WO-2007079930-A1 SUBSTITUTED CYCLOHEXYLMETHYL DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO disclosed