SCHEMBL23153751

SCHEMBL23153751

CP(C)(=O)c1cc(-c2ncc(F)cn2)ccc1Nc1nc(Cl)ncc1Br

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ZAP70 P43403 1/20 0.34
ALK Q9UM73 2/20 0.34
IGF1R P08069 2/20 0.34
INSR P06213 1/20 0.34
PTK2 Q05397 4/20 0.34
P2RX7 Q99572 4/20 0.32
CDK7 P50613 1/20 0.31
CDK9 P50750 1/20 0.31
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23154199 0.91 EGFR (0.39) EGFRMEN1KMT2AALKIGF1R
SCHEMBL23153748 0.89 EGFR (0.41) EGFRMEN1KMT2AALKIGF1R
SCHEMBL23154147 0.88 INSR (0.38) EGFRMEN1KMT2AZAP70ALK
SCHEMBL23154332 0.88 EGFR (0.37) EGFRMEN1KMT2AALKIGF1R
SCHEMBL23154217 0.88 MEN1 (0.40) EGFRMEN1KMT2AALKIGF1R
SCHEMBL24179110 0.87 ALK (0.42) EGFRMEN1KMT2AZAP70ALK
SCHEMBL29977264 0.87 ALK (0.42) EGFRMEN1KMT2AZAP70ALK
SCHEMBL23153980 0.86 MEN1 (0.39) EGFRMEN1KMT2AALKIGF1R
SCHEMBL23154083 0.85 ZAP70 (0.40) EGFRMEN1KMT2AZAP70ALK
SCHEMBL23153875 0.84 EGFR (0.42) EGFRMEN1KMT2AZAP70ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021057882-A1 EGFR INHIBITOR, COMPOSITION AND PREPARATION METHOD THEREFOR 贝达药业股份有限公司 2021-04-01 WO disclosed