SCHEMBL23166300

SCHEMBL23166300

CC(=O)N[C@H]1CCN(C2CCC(N)CC2)C1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
OGFRL1 Q5TC84 2/20 0.38
SLC6A5 Q9Y345 4/20 0.37
CHRM1 P11229 3/20 0.37
AKT1 P31749 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
LTA4H P09960 1/20 0.35
SIGMAR1 Q99720 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14303556 0.85 CHRM1 (0.40) SLC6A5CHRM1HRH3SIGMAR1
SCHEMBL8278776 0.83 SLC6A5 (0.49) CA1CA2CA12CA9OPRM1
SCHEMBL23166392 0.83 SMYD3 (0.41) CHRM1HRH3SIGMAR1
SCHEMBL10076724 0.83 CHRM1 (0.40) CA1CA2CA12CA9OPRM1
SCHEMBL13207164 0.82 EPHX2 (0.50) CA1CA2CA12CA9
SCHEMBL30528703 0.81 CA1 (0.54) CA1CA2CA12CA9CHRM1
SCHEMBL30636651 0.81 CA1 (0.54) CA1CA2CA12CA9CHRM1
SCHEMBL12332584 0.81 POLB (0.44) CA1CA2CA12CA9OPRM1
SCHEMBL8256972 0.79 HRH3 (0.53) CA1CA2CA12CA9HRH3
SCHEMBL30636641 0.77 CA1 (0.53) CA1CA2CA12CA9CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210094912-A1 INDOLE DERIVATIVES AS EFFLUX PUMP INHIBITORS RUTGERS, THE STATE UNIVERISTY OF NEW JERSEY (US) 2021-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210094912-A1 INDOLE DERIVATIVES AS EFFLUX PUMP INHIBITORS ABCB11, ABCB1, ABCG2 CA1 4562/4885CA2 2331/4885CA12 4536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.