SCHEMBL23175643

SCHEMBL23175643

CNc1cc(-c2ccnc(N)c2)ccc1CC=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CIT O14578 1/20 0.39
AAK1 Q2M2I8 4/20 0.37
PDPK1 O15530 1/20 0.36
ABL1 P00519 1/20 0.34
ROCK2 O75116 2/20 0.34
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
IKBKE Q14164 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
LARS1 Q9P2J5 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23175728 0.77 GSK3B (0.37)
SCHEMBL23175609 0.77 HTR6 (0.48) KDM4EMEN1KMT2A
SCHEMBL26012018 0.77 EGLN1 (0.35) ABL1
SCHEMBL23176011 0.72 CHRM1 (0.43) DYRK1A
SCHEMBL23176006 0.69 MAP2K3 (0.38) AAK1
SCHEMBL10528461 0.68 MAPT (0.35) MEN1KMT2A
SCHEMBL30337203 0.68 DYRK1A (0.70) DYRK1AMKNK1MKNK2CITAAK1
SCHEMBL4402187 0.68 DYRK1A (0.63) DYRK1AMKNK1MKNK2AAK1PDPK1
SCHEMBL30935767 0.68 DYRK1A (0.63) DYRK1AMKNK1MKNK2AAK1PDPK1
SCHEMBL8319877 0.68 DYRK1A (0.51) DYRK1AMKNK1MKNK2AAK1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021061053-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (A*STAR) (SG) 2021-04-01 WO disclosed