SCHEMBL23183201

SCHEMBL23183201

COc1ccc2c(c1)N=CCC2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.41
DRD2 P14416 4/20 0.41
DRD3 P35462 4/20 0.41
DRD1 P21728 3/20 0.41
DRD5 P21918 3/20 0.41
BCL2 P10415 1/20 0.40
CHRNA7 P36544 1/20 0.39
CYP11B2 P19099 3/20 0.39
CYP11B1 P15538 1/20 0.39
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
DRD4 P21917 1/20 0.37
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
HTR5A P47898 1/20 0.37
CYP19A1 P11511 2/20 0.37
METAP1 P53582 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20896943 0.86 MPO (0.45) MPODRD2DRD3DRD1DRD5
SCHEMBL7934329 0.76 PARP10 (0.33) CYP11B2HTR5ACYP19A1METAP1
SCHEMBL22900627 0.72 MEN1 (0.38) DRD3DRD1CA2
SCHEMBL29809365 0.72 MEN1 (0.38) DRD3DRD1CA2
SCHEMBL10509271 0.72 PARP1 (0.33) CYP11B2HTR2AHTR2CHTR2BHTR5A
SCHEMBL29531917 0.72 HTR2A (0.38) HTR2AHTR2CHTR2BHTR5A
SCHEMBL16368593 0.71 NPSR1 (0.39)
SCHEMBL3657236 0.71 DRD1 (0.41) DRD2DRD3DRD1DRD5BCL2
SCHEMBL17026922 0.70 BCL2 (0.42) DRD2DRD3DRD1DRD5BCL2
SCHEMBL31022888 0.70 CHRNB2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3798214-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR Vertex Pharmaceuticals Incorporated (US) 2021-03-31 EP disclosed