SCHEMBL23197862

SCHEMBL23197862

C=N/C(Nc1cccc(C(F)F)c1)=C(C=N)\C(C)=N/CC

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDR P35968 1/20 0.33
MAPK14 Q16539 1/20 0.33
TNNI3K Q59H18 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
TSHR P16473 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TOP2A P11388 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23197786 0.74 KDR (0.36) KDM4EMEN1KMT2AKDRMAPK14
SCHEMBL23197819 0.73 MEN1 (0.33) MEN1KMT2AKDRMAPK14TNNI3K
SCHEMBL23197816 0.70 GRIN2D (0.38) MEN1KMT2AKDRMAPK14TNNI3K
SCHEMBL23198944 0.70 TP53 (0.46) KDM4EMEN1KMT2A
SCHEMBL23198668 0.65 NOS3 (0.35) MEN1KMT2AGRIN2DGRIN3BGRIN1
SCHEMBL23198132 0.64 GRIN2D (0.36) KDM4EMEN1KMT2AKDRMAPK14
SCHEMBL23197827 0.64
SCHEMBL19962841 0.63 GRIN2D (0.50) KDM4EMEN1KMT2AKDRGRIN2D
SCHEMBL17762845 0.62 TDO2 (0.40) KDM4EMEN1KMT2AKDRMAPK14
SCHEMBL19232616 0.62 TDO2 (0.37) MEN1KMT2AKDRMAPK14TNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021064077-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES AS IRAK4 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2021-04-08 WO disclosed