SCHEMBL232125

SCHEMBL232125

CC(=N)N[C@@H](CCCN)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 4/20 0.51
SLC6A5 Q9Y345 1/20 0.43
GNPAT O15228 2/20 0.42
CPB2 Q96IY4 5/20 0.40
NOD1 Q9Y239 2/20 0.39
GSR P00390 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
SIRT6 Q8N6T7 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
RNPEP Q9H4A4 1/20 0.37
RIMKLA Q8IXN7 1/20 0.37
NAALAD2 Q9Y3Q0 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
ALOX15 P16050 1/20 0.37
NFKB1 P19838 1/20 0.37
PTGS2 P35354 1/20 0.37
THPO P40225 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL867577 1.00 FOLH1 (0.51) FOLH1SLC6A5GNPATCPB2NOD1
SCHEMBL866580 1.00 FOLH1 (0.51) FOLH1SLC6A5GNPATCPB2NOD1
Hydrochloric Acid SCHEMBL1982441 0.98 FOLH1 (0.50) FOLH1SLC6A5GNPATCPB2NOD1
Hydrochloric Acid SCHEMBL1982438 0.98 FOLH1 (0.50) FOLH1SLC6A5GNPATCPB2NOD1
SCHEMBL45765 0.95 FOLH1 (0.58) FOLH1SLC6A5GNPATCPB2GSR
SCHEMBL214641 0.95 FOLH1 (0.58) FOLH1SLC6A5GNPATCPB2GSR
Hydrochloric Acid SCHEMBL2166126 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
Acetic Acid SCHEMBL268740 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
Hydrochloric Acid SCHEMBL15914484 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
SCHEMBL159460 0.85 GNPAT (0.55) FOLH1SLC6A5GNPATCPB2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 488 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230309521-A1 NOVEL METHOD FOR PREPARING ANIMAL MODEL OF CEREBROVASCULAR DISEASE AND METHOD FOR PRODUCING ANIMAL HAVING SMALL INDIVIDUAL DIFFERENCE IN SUSCEPTIBILITY TO CEREBROVASCULAR DISEASE ONSET BY USING ANIMAL MODEL FOR CEREBROVASCULAR DISEASE PREPARED THEREBY DONGGUK UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2023-10-05 US claimed
EP-4197323-A1 NOVEL METHOD FOR PREPARING ANIMAL MODEL OF CEREBROVASCULAR DISEASE AND METHOD FOR PRODUCING ANIMAL HAVING SMALL INDIVIDUAL DIFFERENCE IN SUSCEPTIBILITY TO CEREBROVASCULAR DISEASE ONSET BY USING ANIMAL MODEL FOR CEREBROVASCULAR DISEASE PREPARED THEREBY Dongguk University Industry-Academic Cooperation Foundation (KR) 2023-06-21 EP claimed
US-20210205468-A1 SYNTHETIC MULTIDOMAIN PEPTIDE BIOMATERIALS THAT INHIBIT INDUCIBLE NITRIC OXIDE SYNTHASE WILLIAM MARSH RICE UNIVERSITY (US) 2021-07-08 US claimed
US-20130130263-A1 GAMETES SEPARATION METHODS, COMPOSITIONS AND USES THEREOF ASSISTANCE PUBLIQUE - HOPITAUX DE PARIS (FR) 2013-05-23 US claimed
EP-2539434-A1 GAMETES SEPARATION METHODS, COMPOSITIONS AND USES THEREOF Assistance Publique - Hôpitaux de Paris (FR) 2013-01-02 EP claimed
US-20120076859-A1 Targeted Lung Delivery of Citrulline and/or Another Nitric Oxide Precursor and a Method for Treatment of Pulmonary Deficiency of Nitric Oxide in Cystic Fibrosis and Other Pulmonary Diseases ACTIVAERO GMBH (DE) 2012-03-29 US claimed
WO-2011104336-A1 GAMETES SEPARATION METHODS, COMPOSITIONS AND USES THEREOF ASSISTANCE PUBLIQUE - HÔPITAUX DE PARIS (FR) 2011-09-01 WO claimed
EP-2361967-A1 Gametes separation methods, compositions and uses thereof Assistance Publique - Hôpitaux de Paris (FR) 2011-08-31 EP claimed
JP-4579349-B2 2010-11-10 JP claimed
WO-2005105065-A2 THIAZOLE-BASED NITRIC OXIDE DONORS FOR TREATING INFLAMMATORY BOWEL DISEASES RENOPHARM LTD. (IL) 2005-11-10 WO claimed
WO-1996002241-A9 USE OF NITROGEN OXIDE SPECIES AND ADDUCTS TO INHIBIT SKELETAL MUSCLE CONTRACTION 1996-02-29 WO claimed
WO-1996002268-A1 INHIBITION OF VIRUS BY NITRIC OXIDE BRIGHAM AND WOMEN'S HOSPITAL (US) 1996-02-01 WO claimed
WO-1996002241-A1 USE OF NITROGEN OXIDE SPECIES AND ADDUCTS TO INHIBIT SKELETAL MUSCLE CONTRACTION DUKE UNIVERSITY (US) 1996-02-01 WO claimed
US-5449688-A Nitric oxide synthase inhibitor or scavenger THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-09-12 US claimed
EP-0603335-A4 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE. US HEALTH (US) 1995-07-05 EP claimed
WO-1995014465-A2 METHODS FOR AMELIORATION OF IMMUNODEFICIENCY VIRUS INDUCED NEURODEGENERATION BY COVERING NITRIC OXIDE OR SUPEROXIDE CONCENTRATION THE JOHNS HOPKINS UNIVERSITY (US) 1995-06-01 WO claimed
WO-1995013805-A1 USE OF NITRIC OXIDE SYNTHASE INHIBITORS IN THE TREATMENT OF AUTOIMMUNE DISEASES DUKE UNIVERSITY MEDICAL CENTER (US) 1995-05-26 WO claimed
EP-0603335-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-06-29 EP claimed
US-5225440-A ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-07-06 US claimed
WO-1993005775-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-04-01 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210205468-A1 SYNTHETIC MULTIDOMAIN PEPTIDE BIOMATERIALS THAT INHIBIT INDUCIBLE NITRIC OXIDE SYNTHASE STING1, CGAS, GMPS FOLH1 1471/4885SLC6A5 4316/4885GNPAT 4260/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.