SCHEMBL866580

SCHEMBL866580

CC(=N)NC(CCCN)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 4/20 0.51
SLC6A5 Q9Y345 1/20 0.43
GNPAT O15228 2/20 0.42
CPB2 Q96IY4 5/20 0.40
NOD1 Q9Y239 2/20 0.39
GSR P00390 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
SIRT6 Q8N6T7 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
RNPEP Q9H4A4 1/20 0.37
RIMKLA Q8IXN7 1/20 0.37
NAALAD2 Q9Y3Q0 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
ALOX15 P16050 1/20 0.37
NFKB1 P19838 1/20 0.37
PTGS2 P35354 1/20 0.37
THPO P40225 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL232125 1.00 FOLH1 (0.51) FOLH1SLC6A5GNPATCPB2NOD1
SCHEMBL867577 1.00 FOLH1 (0.51) FOLH1SLC6A5GNPATCPB2NOD1
Hydrochloric Acid SCHEMBL1982441 0.98 FOLH1 (0.50) FOLH1SLC6A5GNPATCPB2NOD1
Hydrochloric Acid SCHEMBL1982438 0.98 FOLH1 (0.50) FOLH1SLC6A5GNPATCPB2NOD1
SCHEMBL45765 0.95 FOLH1 (0.58) FOLH1SLC6A5GNPATCPB2GSR
SCHEMBL214641 0.95 FOLH1 (0.58) FOLH1SLC6A5GNPATCPB2GSR
Hydrochloric Acid SCHEMBL2166126 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
Acetic Acid SCHEMBL268740 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
Hydrochloric Acid SCHEMBL15914484 0.93 FOLH1 (0.57) FOLH1SLC6A5GNPATCPB2GSR
SCHEMBL159460 0.85 GNPAT (0.55) FOLH1SLC6A5GNPATCPB2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4447916-A1 HAIR CONDITIONING COMPOSITION The Procter & Gamble Company (US) 2024-10-23 EP claimed
WO-2023114680-A1 HAIR CONDITIONING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2023-06-22 WO claimed
US-20230190601-A1 HAIR CONDITIONING COMPOSITION THE PROCTER & GAMBLE COMPANY 2023-06-22 US claimed
US-20120076859-A1 Targeted Lung Delivery of Citrulline and/or Another Nitric Oxide Precursor and a Method for Treatment of Pulmonary Deficiency of Nitric Oxide in Cystic Fibrosis and Other Pulmonary Diseases ACTIVAERO GMBH (DE) 2012-03-29 US claimed
WO-2025122600-A1 COMPOSITIONS AND METHODS FOR TREATING ABERRANT NITROSYLATION CASE WESTERN RESERVE UNIVERSITY (US) 2025-06-12 WO disclosed
EP-4447916-A1 HAIR CONDITIONING COMPOSITION The Procter & Gamble Company (US) 2024-10-23 EP disclosed
CN-118317761-A Hair conditioning composition 宝洁公司 2024-07-09 CN disclosed
US-20230190601-A1 HAIR CONDITIONING COMPOSITION THE PROCTER & GAMBLE COMPANY 2023-06-22 US disclosed
WO-2023114680-A1 HAIR CONDITIONING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2023-06-22 WO disclosed
US-20180161376-A1 COMPOSITIONS AND METHODS FOR NEURONAL DIFFERENTIATION OF CELLS NORTHERN SYDNEY LOCAL HEALTH DISTRICT (AU) 2018-06-14 US disclosed
EP-2308510-B1 Agent for regeneration and/or protection of nerves ONO PHARMACEUTICAL CO (JP) 2016-03-16 EP disclosed
CN-104940126-A Controlled-release otic structure modulating and innate immune system modulating compositions and methods for the treatment of otic disorders OTONOMY INC 2015-09-30 CN disclosed
EP-0750906-A1 DELTA-(S-METHYLISOTHIOUREIDO)-L-NORVALINE AND CEREBROVASCULAR DISORDER REMEDY HAVING NITROGEN MONOXIDE SYNTHASE INHIBITOR ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-01-02 EP disclosed
EP-0718294-A1 2-Amino-1,3-thiazepines and their use as inhibitors of the nitrogene oxide synthase HOECHST AKTIENGESELLSCHAFT (DE) 1996-06-26 EP disclosed
EP-0713704-A1 2-Amino-1,3-thiazines as nitric oxide synthase inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1996-05-29 EP disclosed
EP-0603335-A4 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE. US HEALTH (US) 1995-07-05 EP disclosed
WO-1994023038-A1 INDUCIBLE NITRIC OXIDE SYNTHASE AND GENE THEREFOR THE WELLCOME FOUNDATION LIMITED (GB) 1994-10-13 WO disclosed
EP-0603335-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-06-29 EP disclosed
US-5225440-A ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-07-06 US disclosed
WO-1993005775-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-04-01 WO disclosed