SCHEMBL23212526

SCHEMBL23212526

NC(=O)C1Cc2ccncc2N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
GAA P10253 1/20 0.42
NAMPT P43490 2/20 0.41
SIRT3 Q9NTG7 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
NNMT P40261 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
SARM1 Q6SZW1 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT6 Q8N6T7 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT5 Q9NXA8 1/20 0.33
SIRT4 Q9Y6E7 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
KDM6B O15054 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31092717 0.89 MAPT (0.44) MAPTGAANAMPTSIRT3TDP1
SCHEMBL17541892 0.84 SMYD3 (0.39) MAPTGAANAMPTSIRT3TDP1
Hydrochloric Acid SCHEMBL21545777 0.83 SMYD3 (0.39) NAMPTSIRT3TDP1NNMTCHRNB2
SCHEMBL13660486 0.79 NAMPT (0.42) MAPTGAANAMPTHRH4TSHR
SCHEMBL10742930 0.76 GAA (0.71) MAPTGAA
SCHEMBL30900484 0.76 GAA (0.71) MAPTGAA
SCHEMBL2266601 0.76 GAA (0.71) MAPTGAA
Hydrochloric Acid SCHEMBL28262901 0.75 GAA (0.69) MAPTGAA
SCHEMBL22411406 0.73 MAPT (0.41) MAPTGAANAMPTCHRNB2CHRNA4
SCHEMBL13271647 0.72 CHRNB2 (0.35) MAPTGAANNMTSIRT6CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021068755-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发股份有限公司 2021-04-15 WO disclosed