SCHEMBL23222258

SCHEMBL23222258

COc1cccc(CC2CN(C=O)CCN2)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.45
HTR1A P08908 1/20 0.45
EED O75530 2/20 0.44
SIGMAR1 Q99720 3/20 0.44
CHRM4 P08173 2/20 0.43
DRD2 P14416 2/20 0.43
HTR7 P34969 2/20 0.43
SLC6A2 P23975 1/20 0.41
ROCK2 O75116 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
CMA1 P23946 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10388535 0.82 POLB (0.49) SLC6A4SLC6A2
SCHEMBL19049075 0.80 CCR3 (0.51) SLC6A4HTR1AEEDSIGMAR1KDM4E
SCHEMBL4281534 0.80 CCR3 (0.49) SLC6A4HTR1AEEDSIGMAR1KDM4E
SCHEMBL13858982 0.80 SLC6A4 (0.47) SLC6A4HTR1AEEDSIGMAR1CHRM4
SCHEMBL19002806 0.78 CCR3 (0.47) EEDSIGMAR1KDM4EALDH1A1
SCHEMBL21169224 0.77 CCR3 (0.47) EEDSIGMAR1KDM4EALDH1A1
SCHEMBL6132670 0.76 CCR3 (0.45) EEDROCK2KDM4EALDH1A1
SCHEMBL13705102 0.76 CCR3 (0.45) EEDROCK2KDM4EALDH1A1
SCHEMBL3154073 0.74 EED (0.63) SLC6A4HTR1AEEDCHRM4DRD2
SCHEMBL18668 0.73 ALDH1A1 (0.55) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3642209-B1 COMPOUNDS THAT INTERACT WITH THE RAS SUPERFAMILY FOR THE TREATMENT OF CANCERS, INFLAMMATORY DISEASES, RASOPATHIES, AND FIBROTIC DISEASE SHY Therapeutics LLC (US) 2023-11-29 EP disclosed
EP-3394056-B1 COMPOUNDS FOR THE TREATMENT OF CANCER AND INFLAMMATORY DISEASE SHY Therapeutics LLC (US) 2021-04-14 EP disclosed