SCHEMBL23232249

SCHEMBL23232249

COc1cccc(F)c1C1(N)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.42
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MAPK1 P28482 2/20 0.38
ACHE P22303 2/20 0.38
ALDH1A1 P00352 2/20 0.38
ADRA2B P18089 1/20 0.38
PTGS1 P23219 1/20 0.38
KMT2A Q03164 1/20 0.37
HPGD P15428 2/20 0.37
NPC1 O15118 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6904575 0.81 HTR5A (0.34)
SCHEMBL23231438 0.78 SIGMAR1 (0.39) NFE2L2TDP1CA12CA1CA2
SCHEMBL31614233 0.77 SIGMAR1 (0.41) NFE2L2TDP1L3MBTL1CA12CA1
SCHEMBL23231270 0.75 HTR2A (0.37)
SCHEMBL23232571 0.74 KRAS (0.34) NFE2L2KMT2A
SCHEMBL18769733 0.73
SCHEMBL1132825 0.72 SIGMAR1 (0.51) TDP1L3MBTL1CA12CA1CA2
SCHEMBL31159059 0.72 HTR5A (0.33)
Hydrochloric Acid SCHEMBL18742474 0.71
SCHEMBL108534 0.71 TDP1 (0.48) NFE2L2TDP1L3MBTL1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021071843-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS Pipeline Therapeutics, Inc. (US) 2021-04-15 WO disclosed