SCHEMBL2324324

SCHEMBL2324324

C=CCN(CC=C)C(=O)OCc1ccccc1.O=C(Cl)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
HCAR2 Q8TDS4 1/20 0.45
CCR6 P51684 1/20 0.45
PAX8 Q06710 1/20 0.45
KMT2A Q03164 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
LMNA P02545 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TGM2 P21980 1/20 0.39
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
CA12 O43570 1/20 0.38
AKR1B10 O60218 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL541750 0.93 HCAR2 (0.51) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL651119 0.87 CCR6 (0.49) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL15297836 0.86 HCAR2 (0.45) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL4690235 0.85 HCAR2 (0.47) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL21573938 0.84 ALDH1A1 (0.47) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL1517791 0.84 HCAR2 (0.46) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL650849 0.83 HCAR2 (0.43) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL650850 0.83 HCAR2 (0.43) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL19216108 0.83 SIGMAR1 (0.44) ALDH1A1HCAR2CCR6PAX8KMT2A
SCHEMBL6899637 0.83 HCAR2 (0.43) ALDH1A1HCAR2CCR6PAX8KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356125-A1 DERIVATIVES OF OXABISPIDINE AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS Targacept, Inc. (US) 2011-08-17 EP disclosed
WO-2010002971-A1 DERIVATIVES OF OXABISPIDINE AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-01-07 WO disclosed