SCHEMBL2324809

SCHEMBL2324809

N=C(NO)c1ccc(OCC(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 5/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
HTT P42858 4/20 0.40
NPSR1 Q6W5P4 3/20 0.40
LMNA P02545 3/20 0.40
PAX8 Q06710 2/20 0.40
ALDH1A1 P00352 3/20 0.39
PRSS1 P07477 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP17A1 P05093 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP1A2 P05177 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
S1PR2 O95136 1/20 0.37
S1PR4 O95977 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23578263 0.82 PRSS1 (0.45) PRSS1TMPRSS2
SCHEMBL23068921 0.81 KDM4E (0.46) KDM4EMAPTHTTPRSS1
SCHEMBL18104847 0.80 PRSS1 (0.41) PRSS1TMPRSS2
SCHEMBL548439 0.78 PRSS1 (0.60) PRSS1L3MBTL1GAATMPRSS2
SCHEMBL549185 0.78 TMPRSS2 (0.60) PRSS1L3MBTL1TMPRSS2
SCHEMBL498377 0.77 ALDH1A1 (0.56) SMN1; SMN2NPC1RAB9AKDM4EMAPT
Pentamidine Dao SCHEMBL548448 0.77 PRMT1 (0.61) PRSS1L3MBTL1GAATMPRSS2
SCHEMBL2323023 0.77 EPHX2 (0.46) NPC1RAB9AKDM4EMAPTL3MBTL1
SCHEMBL20946216 0.76 MAPK14 (0.47) KDM4EMAPTMEN1KMT2ALMNA
SCHEMBL409427 0.75 NR1I2 (0.53) SMN1; SMN2MAPTALDH1A1PRSS1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356112-A1 HETEROAROMATIC COMPOUNDS FOR USE AS HIF INHIBITORS Bayer Schering Pharma Aktiengesellschaft (DE) 2011-08-17 EP disclosed
WO-2010054764-A1 HETEROAROMATIC COMPOUNDS FOR USE AS HIF INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-05-20 WO disclosed