SCHEMBL23258154

SCHEMBL23258154

CCOC(=O)/C=C/c1cn(COCC[Si](C)(C)C)c(=O)c(N2CCS(=O)(=O)CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.33
KLKB1 P03952 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
RECQL P46063 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23257963 0.91 RXFP1 (0.35) DGAT1KLKB1NPC1RAB9A
SCHEMBL21564465 0.89 ALDH1A1 (0.35) DGAT1KLKB1
SCHEMBL21553173 0.89 KLKB1 (0.34) KLKB1
SCHEMBL26031543 0.83 PFKFB3 (0.36) DGAT1KLKB1NPC1RAB9A
SCHEMBL21553045 0.80 DGAT1 (0.35) DGAT1KLKB1
SCHEMBL21552828 0.79 KLKB1 (0.35) DGAT1KLKB1
SCHEMBL21552892 0.77 DGAT1 (0.38) DGAT1KLKB1
SCHEMBL21552990 0.74 DGAT1 (0.34) DGAT1KLKB1
SCHEMBL21552924 0.74
SCHEMBL26031607 0.73 DGAT1 (0.34) DGAT1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230250090-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE IMAGO BIOSCIENCES INC (US) 2023-08-10 US disclosed
US-20230250090-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE IMAGO BIOSCIENCES INC (US) 2023-08-10 US disclosed
US-11578059-B2 KDM1A inhibitors for the treatment of disease Imago Biosciences. Inc. (US) 2023-02-14 US disclosed
US-20210115023-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE IMAGO BIOSCIENCES, INC. 2021-04-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230250090-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE KDM1B, KDM1A, KDM2A DGAT1 2741/4885KLKB1 1359/4885NPC1 4463/4885
US-20210115023-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE KDM1A, KDM1B, KDM2A DGAT1 2605/4885KLKB1 1280/4885NPC1 4422/4885
US-11578059-B2 KDM1A inhibitors for the treatment of disease KDM1B, KDM1A, KDM2A DGAT1 2741/4885KLKB1 1359/4885NPC1 4463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.