SCHEMBL23262015

SCHEMBL23262015

C=CN(C)c1c(C)ncn(CC#N)c1=O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.40
ALDH1A1 P00352 5/20 0.39
MEN1 O00255 3/20 0.39
POLB P06746 3/20 0.39
KMT2A Q03164 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 2/20 0.37
PDE4A P27815 1/20 0.36
ADORA2A P29274 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PKM P14618 1/20 0.35
CSNK2A1 P68400 1/20 0.33
CYP1A2 P05177 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CYP17A1 P05093 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23718388 0.72
SCHEMBL17008902 0.65 CSNK2A1 (0.42) ADORA2BALDH1A1MEN1POLBKMT2A
SCHEMBL17020156 0.64 ADORA2B (0.41) ADORA2BALDH1A1MEN1POLBKMT2A
SCHEMBL23246540 0.62 ADORA2B (0.52) ADORA2BALDH1A1MEN1POLBKMT2A
SCHEMBL17008879 0.62 LMNA (0.42) ADORA2BALDH1A1MEN1POLBKMT2A
SCHEMBL10652515 0.57 ADORA2B (1.00) ADORA2BALDH1A1POLBPDE4AADORA2A
SCHEMBL1956056 0.57
SCHEMBL6362430 0.57 KDM4E (0.43) ALDH1A1MEN1POLBKMT2AL3MBTL1
SCHEMBL20888904 0.56 ADORA2B (0.36) ADORA2BALDH1A1MEN1POLBKMT2A
SCHEMBL27404798 0.54 ADORA2B (0.34) ADORA2BPOLBADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021074198-A1 NOVEL TETRAZOLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-04-22 WO disclosed