SCHEMBL2331266

SCHEMBL2331266

CC(=O)c1ccc(Cn2nc(C(N)=O)c(-c3nc(C(=O)O)c(-c4cccc(Cl)c4)o3)n2)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.45
RXRA P19793 2/20 0.38
RXRB P28702 2/20 0.38
RXRG P48443 2/20 0.38
NR4A2 P43354 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AVPR1B P47901 2/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
SLC9A1 P19634 2/20 0.35
MDM2 Q00987 3/20 0.35
PDE4B Q07343 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2328930 0.91 HCRTR1 (0.44) IKBKBRXRARXRBRXRGNR4A2
SCHEMBL2323238 0.90 IKBKB (0.40) IKBKBNR4A2HCRTR1HCRTR2KDM4E
SCHEMBL2332690 0.90 NR4A1 (0.37) IKBKBNR4A2HCRTR1HCRTR2SLC9A1
SCHEMBL2327523 0.90 IKBKB (0.41) IKBKBRXRARXRBRXRGMEN1
SCHEMBL2327731 0.88 RXRA (0.41) IKBKBRXRARXRBRXRGMEN1
SCHEMBL2327570 0.88 LRRK2 (0.36) IKBKBHCRTR1HCRTR2KDM4EALDH1A1
SCHEMBL2327049 0.88 IKBKB (0.48) IKBKBRXRARXRBKMT2ASLC9A1
SCHEMBL2328920 0.88 IKBKB (0.35) IKBKBKMT2AHCRTR1HCRTR2ALDH1A1
SCHEMBL1704456 0.87 IKBKB (0.41) IKBKBRXRARXRBRXRGNR4A2
SCHEMBL2328104 0.86 HCRTR1 (0.36) IKBKBRXRARXRBKMT2AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP claimed
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP disclosed