SCHEMBL23325964

SCHEMBL23325964

COc1ccc(C2(C#N)CCNCC2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 19/20 0.53
PDE4A P27815 18/20 0.53
PDE4C Q08493 18/20 0.53
PDE4D Q08499 18/20 0.53
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL77276 0.89 PDE4B (0.59) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL13761090 0.87 OPRM1 (0.47) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL13761156 0.87 PDE4B (0.44) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL13526162 0.86 PDE4B (0.73) PDE4BPDE4APDE4CPDE4D
SCHEMBL2827366 0.86 PDE4B (0.59) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL558312 0.86 MEN1 (0.61) PDE4BPDE4APDE4CPDE4DMEN1
Hydrochloric Acid SCHEMBL3181049 0.85 PDE4B (0.72) PDE4BPDE4APDE4CPDE4D
SCHEMBL558606 0.84 MEN1 (0.60) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL14544227 0.84 PDE4B (0.42) PDE4BPDE4APDE4CPDE4DMEN1
SCHEMBL7381516 0.81 PDE4B (0.75) PDE4BPDE4APDE4CPDE4DMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021083328-A1 POLYSUBSTITUTED ISOINDOLINE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 中国科学院上海药物研究所 2021-05-06 WO disclosed