SCHEMBL23328829

SCHEMBL23328829

CC(C)CN1C(=O)COCC1C

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 6/20 0.45
CACNA1B Q00975 1/20 0.34
POLB P06746 1/20 0.33
PER2 O15055 4/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14376300 0.74 PIK3CD (0.66) PIK3CD
SCHEMBL22854583 0.72 SIGMAR1 (0.41) POLB
SCHEMBL24391283 0.72 NSD2 (0.32) NOTUM
SCHEMBL9654559 0.71 GBA1 (0.41) POLB
SCHEMBL19231898 0.71 PRMT5 (0.51) PER2
SCHEMBL22833754 0.70 BRD4 (0.36)
SCHEMBL1008150 0.70 P2RX7 (0.46)
SCHEMBL22854580 0.70 PLK1 (0.36) POLB
SCHEMBL1189963 0.70 P2RX7 (0.46)
SCHEMBL12213138 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230012600-A1 BRIDGED CYCLOFORMYLPYRIDINE DERIVATIVES AND USES THEREOF BROADENBIO CO., LTD. (CN) 2023-01-19 US disclosed
WO-2021083011-A1 BRIDGED CYCLOFORMYLPYRIDINE DERIVATIVE AND USE THEREOF 北京伯汇生物技术有限公司 2021-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230012600-A1 BRIDGED CYCLOFORMYLPYRIDINE DERIVATIVES AND USES THEREOF FGFR4, FGFR1, FGFR3 PIK3CD 815/4885CACNA1B 2823/4885POLB 1151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.