SCHEMBL2334680

SCHEMBL2334680

CC(Cl)C(C#N)c1ccc(C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.43
ESR2 Q92731 3/20 0.43
TSHR P16473 2/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
ALOX15 P16050 1/20 0.39
RXRA P19793 3/20 0.39
RXRB P28702 3/20 0.39
NR1H4 Q96RI1 1/20 0.39
ANPEP P15144 1/20 0.39
RXRG P48443 1/20 0.38
SRD5A2 P31213 1/20 0.38
LMNA P02545 3/20 0.37
ALPG P10696 2/20 0.37
HPGD P15428 2/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2335804 0.81 ANPEP (0.45) ESR1ESR2ALDH1A1SMN1; SMN2RXRA
SCHEMBL7302128 0.78 TSHR (0.48) TSHRTP53KMT2AALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL9695884 0.77 TSHR (0.46) TSHRTP53KMT2AALDH1A1SMN1; SMN2
SCHEMBL5124953 0.75 TSHR (0.55) TSHRTP53KMT2AALDH1A1SMN1; SMN2
Terephthalic Acid SCHEMBL9017249 0.74 TSHR (0.67) TSHRTP53KMT2AALDH1A1SMN1; SMN2
SCHEMBL15543858 0.72 TSHR (0.50) TSHRTP53KMT2AALDH1A1SMN1; SMN2
SCHEMBL28932021 0.71 MAPT (0.47) ESR1ESR2TSHRTP53KMT2A
SCHEMBL31192242 0.71 TSHR (0.60) TSHRTP53KMT2AALDH1A1SMN1; SMN2
SCHEMBL8154043 0.71 TSHR (0.60) TSHRTP53ALDH1A1SMN1; SMN2ALOX15
SCHEMBL105270 0.71 RXRA (0.62) TSHRTP53KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358689-A1 Benzothiazole derivatives as anticancer agents Takeda Pharmaceutical Company Limited (JP) 2011-08-24 EP disclosed
WO-2010064722-A1 BENZOTHIAZOLE DERIVATIVES AS ANTICANCER AGENTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-10 WO disclosed