SCHEMBL23349338

SCHEMBL23349338

Cc1ncc2ccccccccc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.47
KDM4E B2RXH2 2/20 0.45
GPR3 P46089 2/20 0.45
EGFR P00533 1/20 0.45
CYP2A6 P11509 1/20 0.45
HTR3A P46098 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
PDE10A Q9Y233 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 2/20 0.42
GLA P06280 1/20 0.42
ACHE P22303 1/20 0.42
STAT3 P40763 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL196151 0.98 CYP1A2 (0.48) CYP1A2KDM4EGPR3EGFRCYP2A6
Water SCHEMBL27373628 0.95 CYP1A2 (0.47) CYP1A2KDM4EGPR3EGFRCYP2A6
Formaldehyde SCHEMBL28015338 0.91 CYP1A2 (0.44) CYP1A2KDM4EGPR3EGFRCYP2A6
Piperazine SCHEMBL27739524 0.86 HTR3A (0.42) CYP1A2KDM4EGPR3EGFRCYP2A6
SCHEMBL12033738 0.78 CYP1A2 (0.52) CYP1A2KDM4EGPR3CYP2A6ALDH1A1
SCHEMBL30059022 0.76 CYP1A2 (0.45) CYP1A2KDM4EGPR3PDE10AALDH1A1
SCHEMBL17532748 0.75 LMNA (0.61) CYP1A2KDM4EGPR3CYP2A6ALDH1A1
SCHEMBL21959296 0.75 MEN1 (0.42) KDM4EGPR3CYP2A6PDE10AALDH1A1
SCHEMBL8404379 0.74 CYP1A2 (0.42) CYP1A2KDM4EGPR3CYP2A6ALDH1A1
SCHEMBL30527184 0.73 CYP1A2 (0.60) CYP1A2KDM4EGPR3EGFRCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210139482-A1 SUBSTITUTED 1,2-DIHYDRO-3H-PYRAZOLO[3,4-D]PYRIMIDIN-3-ONES RECURIUM IP HOLDINGS, LLC 2021-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210139482-A1 SUBSTITUTED 1,2-DIHYDRO-3H-PYRAZOLO[3,4-D]PYRIMIDIN-3-ONES MKI67, BRCA1, CCNI CYP1A2 361/4885KDM4E 2533/4885GPR3 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.