SCHEMBL23356302

SCHEMBL23356302

O=C(Oc1ccncc1)c1cc(C(F)(F)F)cnc1Oc1ccc(OC(F)(F)F)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
ATM Q13315 1/20 0.47
LIPE Q05469 1/20 0.43
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 5/20 0.41
FFAR1 O14842 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
SCN9A Q15858 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
HPGD P15428 1/20 0.37
CSF1R P07333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31344110 0.86 SMN1; SMN2 (0.48) KMT2AATMLIPELMNASMN1; SMN2
SCHEMBL23356328 0.86 SMN1; SMN2 (0.48) KMT2AATMLIPELMNASMN1; SMN2
SCHEMBL23356327 0.80 KMT2A (0.53) KMT2AATMSMN1; SMN2
SCHEMBL29737621 0.80 KMT2A (0.53) KMT2AATMSMN1; SMN2
SCHEMBL31344113 0.79 KMT2A (0.51) KMT2AATMSMN1; SMN2RAB9ASCN9A
SCHEMBL31344025 0.79 KMT2A (0.51) KMT2AATMSMN1; SMN2
SCHEMBL23356237 0.79 KMT2A (0.51) KMT2AATMSMN1; SMN2
SCHEMBL23356260 0.79 KMT2A (0.51) KMT2AATMSMN1; SMN2RAB9ASCN9A
SCHEMBL23356269 0.78 KMT2A (0.53) KMT2AATMSMN1; SMN2
SCHEMBL23356160 0.78 SORT1 (0.51) KMT2AATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260001861-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 LIEBER INST INC (US) 2026-01-01 US claimed
US-20220227732-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 LIEBER INSTITUTE, INC 2022-07-21 US claimed
EP-3820866-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 Lieber Institute, Inc. (US) 2021-05-19 EP claimed
CN-112689633-A For inhibiting Nav1.8 pyridine carboxamide Compounds 利伯研究所公司 2021-04-20 CN claimed
US-20260001861-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 LIEBER INST INC (US) 2026-01-01 US disclosed
US-12234221-B2 Pyridine carboxamide compounds for inhibiting NAV1.8 LIEBER INSTITUTE, INC. (US) 2025-02-25 US disclosed
US-20220227732-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 LIEBER INSTITUTE, INC 2022-07-21 US disclosed
EP-3820866-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 Lieber Institute, Inc. (US) 2021-05-19 EP disclosed
CN-112689633-A For inhibiting Nav1.8 pyridine carboxamide Compounds 利伯研究所公司 2021-04-20 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220227732-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 SCN8A, SCN1A, SCN2A KMT2A 1228/4885ATM 4626/4885LIPE 4787/4885
US-12234221-B2 Pyridine carboxamide compounds for inhibiting NAV1.8 SCN8A, SCN1A, SCN2A KMT2A 1228/4885ATM 4626/4885LIPE 4787/4885
US-20260001861-A1 PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8 SCN8A, SCN1A, SCN1B KMT2A 2792/4885ATM 4836/4885LIPE 4495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.