SCHEMBL23377685

SCHEMBL23377685

COc1ccc(O[C@H]2CN[C@@H](C)C2)cn1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.47
CHRNA4 P43681 5/20 0.47
CHRNB4 P30926 3/20 0.40
CHRNA3 P32297 3/20 0.40
CHRNA7 P36544 1/20 0.40
CHRM4 P08173 4/20 0.39
OXTR P30559 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23377715 0.82 CHRNB2 (0.45) CHRNB2CHRNA4CHRM4
SCHEMBL23377601 0.82 CHRNB2 (0.45) CHRNB2CHRNA4CHRM4
Hydrochloric Acid SCHEMBL28633579 0.81 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL28645846 0.81 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL31470955 0.81 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL29053972 0.79 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL23377702 0.78 HCRTR1 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL23377547 0.77 CHRNB2 (0.47) CHRNB2CHRNA4
SCHEMBL22666841 0.77 SLC6A4 (0.55) CHRNB2CHRNA4CHRM4
SCHEMBL19050128 0.77 SLC6A4 (0.55) CHRNB2CHRNA4CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021094312-A1 PYRROLIDINE AND BICYCLOHETEROARYL CONTAINING OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2021-05-20 WO disclosed