SCHEMBL23377702

SCHEMBL23377702

Cc1ccc(O[C@H]2CN[C@@H](C)C2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CHRNB2 P17787 3/20 0.32
CHRNA4 P43681 3/20 0.32
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31
HRH3 Q9Y5N1 3/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16716333 0.84 FPR2 (0.39) HCRTR1CHRNB2CHRNA4
SCHEMBL21807911 0.84 TDO2 (0.37) HCRTR1HCRTR2CHRNB2CHRNA4CHRNA7
SCHEMBL21807928 0.84 DGAT1 (0.39) HCRTR1HCRTR2KDM4ECHRNB2CHRNA4
SCHEMBL10078038 0.82 HCRTR1 (0.40) HCRTR1HCRTR2KDM4EALDH1A1HSD17B10
SCHEMBL20323923 0.79 HCRTR2 (0.40) HCRTR1HCRTR2KDM4EALDH1A1HSD17B10
SCHEMBL23377548 0.79 NOS3 (0.31) NOS3NOS2
SCHEMBL23377685 0.78 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL20261372 0.77 HCRTR1 (0.44) HCRTR1HCRTR2KDM4EALDH1A1HSD17B10
SCHEMBL23377711 0.76 NOS3 (0.31) NOS3NOS2
SCHEMBL23167660 0.74 NOS3 (0.38) HCRTR1HCRTR2KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021094312-A1 PYRROLIDINE AND BICYCLOHETEROARYL CONTAINING OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2021-05-20 WO disclosed