SCHEMBL2340969

SCHEMBL2340969

C[C@@H](C(=N)NCCCN(C)C)c1cccc(C(=O)c2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.54
PTGS1 P23219 3/20 0.54
PTGS2 P35354 3/20 0.54
ALDH1A1 P00352 3/20 0.54
CXCR1 P25024 2/20 0.54
CXCR2 P25025 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
LMNA P02545 2/20 0.54
CYP3A4 P08684 2/20 0.54
HPGD P15428 2/20 0.54
RECQL P46063 1/20 0.54
KDM4E B2RXH2 1/20 0.54
MAPK1 P28482 1/20 0.54
PMP22 Q01453 1/20 0.54
SLC22A6 Q4U2R8 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CXCL8 P10145 1/20 0.54
THPO P40225 1/20 0.54
HIF1A Q16665 1/20 0.54
MEN1 O00255 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446061 1.00 MAPT (0.54) MAPTPTGS1PTGS2ALDH1A1CXCR1
Hydrochloric Acid SCHEMBL2336294 0.99 MAPT (0.53) MAPTPTGS1PTGS2ALDH1A1CXCR1
Hydrochloric Acid SCHEMBL2336298 0.99 MAPT (0.53) MAPTPTGS1PTGS2ALDH1A1CXCR1
Hydrochloric Acid SCHEMBL2342127 0.99 MAPT (0.53) MAPTPTGS1PTGS2ALDH1A1CXCR1
SCHEMBL4910072 0.89 GLI1 (0.64) MAPTPTGS1PTGS2ALDH1A1CXCR1
SCHEMBL17889135 0.89 GLI1 (0.64) MAPTPTGS1PTGS2ALDH1A1CXCR1
SCHEMBL11624162 0.85 GLI1 (0.61) MAPTPTGS1PTGS2ALDH1A1CXCR1
Ketoprofen SCHEMBL2286417 0.79 PTGS1 (0.74) MAPTPTGS1PTGS2ALDH1A1CXCR1
SCHEMBL4909390 0.79 GLI1 (0.62) MAPTPTGS1PTGS2ALDH1A1CXCR1
SCHEMBL17192952 0.79 PTGS2 (0.63) MAPTPTGS1PTGS2ALDH1A1CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663960-B1 AMIDINES AND DERIVATIVES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPE SPA (IT) 2011-08-24 EP disclosed