SCHEMBL23442811

SCHEMBL23442811

COOc1c(Cl)cc(-n2nc(C(=O)O)c(=O)[nH]c2=O)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 12/20 0.60
THRB P10828 12/20 0.49
L3MBTL1 Q9Y468 2/20 0.46
CYP2C9 P11712 2/20 0.41
UGT1A1 P22309 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
SLCO1B1 Q9Y6L6 1/20 0.41
ATM Q13315 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C8 P10632 1/20 0.39
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
STAT1 P42224 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
LMNA P02545 1/20 0.36
GRIK1 P39086 1/20 0.36
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36
GRIA3 P42263 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23663177 0.83 THRA (0.61) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL10408308 0.82 THRA (0.55) THRATHRBL3MBTL1ATMKMT2A
SCHEMBL11471529 0.80 THRA (0.54) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL11465964 0.78 THRA (0.58) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL23663471 0.78 THRA (0.60) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL23442810 0.78 THRB (0.52) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL2921588 0.76 THRA (1.00) THRATHRBCYP2C9UGT1A1ABCG2
SCHEMBL23168580 0.76 THRA (0.60) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL23168797 0.76 THRA (0.65) THRATHRBL3MBTL1CYP2C9UGT1A1
SCHEMBL29066220 0.76 THRA (0.55) THRATHRBL3MBTL1CYP2C9UGT1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021104288-A1 1,2,4-TRIAZINE-3,5-DIONE COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 昆药集团股份有限公司 2021-06-03 WO disclosed