SCHEMBL2345331

SCHEMBL2345331

CN(C)CCOc1cc(-c2cnc3[nH]cc(OC(=O)NCC(C)(C)CO)c3n2)cc(N2CCC(C)(C)C2)c1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.38
SYK P43405 6/20 0.34
CYP2D6 P10635 1/20 0.34
KCNH2 Q12809 1/20 0.34
NTRK1 P04629 1/20 0.33
RET P07949 2/20 0.31
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2278401 0.90 SYK (0.41) MAP4K1SYKCYP2D6KCNH2CYP2C9
SCHEMBL2344505 0.87 MAP4K1 (0.36) MAP4K1SYKCYP2D6CYP2C9
SCHEMBL2273339 0.82 JAK3 (0.43) MAP4K1SYKCYP2D6KCNH2CYP2C9
SCHEMBL3063499 0.81 MAP4K1 (0.40) MAP4K1SYKCYP2D6KCNH2NTRK1
SCHEMBL2278409 0.78 SYK (0.38) MAP4K1SYKCYP2D6KCNH2NTRK1
SCHEMBL2348276 0.77 SYK (0.38) MAP4K1SYKCYP2D6KCNH2
SCHEMBL2274314 0.75 SYK (0.41) SYKCYP2D6KCNH2CYP2C9
SCHEMBL2344717 0.74 SYK (0.37) MAP4K1SYKCYP2D6KCNH2CYP2C9
SCHEMBL2350193 0.72 SYK (0.38) MAP4K1SYKCYP2C9
SCHEMBL2351523 0.72 SYK (0.54) SYKCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245033-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed