SCHEMBL2344717

SCHEMBL2344717

CC1(C)CCN(c2cccc(-c3cnc4[nH]cc(OC(=O)NC(C)(C)C)c4n3)c2)C1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SYK P43405 12/20 0.37
CYP2D6 P10635 2/20 0.37
KCNH2 Q12809 1/20 0.37
PRKCI P41743 1/20 0.36
MAP4K1 Q92918 2/20 0.35
ATR Q13535 1/20 0.35
MAPK1 P28482 1/20 0.35
JAK3 P52333 2/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2348276 0.92 SYK (0.38) SYKCYP2D6KCNH2PRKCIMAP4K1
SCHEMBL2349020 0.89 SYK (0.41) SYKCYP2D6KCNH2PRKCIMAP4K1
SCHEMBL2341691 0.88 SYK (0.43) SYKPRKCIMAP4K1JAK3CYP2C9
SCHEMBL2341503 0.88 JAK3 (0.39) SYKPRKCIMAP4K1ATRJAK3
SCHEMBL2349820 0.88 ATR (0.45) PRKCIATRJAK3
SCHEMBL2344505 0.87 MAP4K1 (0.36) SYKCYP2D6PRKCIMAP4K1ATR
SCHEMBL2278920 0.86 SYK (0.50) SYKCYP2D6KCNH2
SCHEMBL2350193 0.84 SYK (0.38) SYKPRKCIMAP4K1ATRMAPK1
SCHEMBL2362648 0.83 JAK3 (0.36) SYKCYP2D6KCNH2MAP4K1ATR
SCHEMBL2343568 0.82 CNR2 (0.40) SYKATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245033-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed