SCHEMBL23471111

SCHEMBL23471111

CC(=O)NCc1cccc(C(=O)NCCN2CCS[C@H](C)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 5/20 0.42
PARP1 P09874 3/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ROCK2 O75116 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DRD4 P21917 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634745 0.81 PARP1 (0.59) CHRM3PARP1CYP2C9CYP2C19HSD17B10
SCHEMBL19634814 0.80 CHRM3 (0.46) CHRM3ROCK2
SCHEMBL23471125 0.79 CYP2C19 (0.65) PARP1CYP2C9CYP2C19
SCHEMBL23471112 0.79 CHRM3 (0.61) CHRM3PARP1
SCHEMBL19634727 0.77 TMEM97 (0.38) CHRM3PARP1CYP2C9CYP2C19TMEM97
SCHEMBL23471004 0.77 PARP1 (0.48) CHRM3PARP1CYP2C9CYP2C19HSD17B10
SCHEMBL23471126 0.77 PARP1 (0.48) PARP1CYP2C9TMEM97HSD17B10
SCHEMBL21015957 0.74 CYP2C9 (0.46) CHRM3PARP1CYP2C9CYP2C19TMEM97
SCHEMBL16380331 0.73 ROCK2 (0.53) CYP2C9HSD17B10ROCK2
SCHEMBL19634640 0.72 LMNA (0.53) PARP1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed