SCHEMBL2353322

SCHEMBL2353322

[c]1nccc(N2CCCCC2)c1-c1cccnn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 7/20 0.49
CDC42BPB Q9Y5S2 7/20 0.49
ROCK2 O75116 6/20 0.49
CDC42BPA Q5VT25 3/20 0.34
OPRK1 P41145 1/20 0.34
METAP1 P53582 2/20 0.34
HPGD P15428 1/20 0.33
DHFR P00374 1/20 0.33
KEAP1 Q14145 1/20 0.33
SMARCA2 P51531 2/20 0.32
SMARCA4 P51532 2/20 0.32
PBRM1 Q86U86 2/20 0.32
NR1I2 O75469 1/20 0.32
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3760229 0.76 KDM4E (0.43) HPGDKEAP1RAB9ANPC1ALDH1A1
SCHEMBL6850968 0.75 KDM4E (0.44) METAP1RAB9ANPC1ALDH1A1MAPK1
SCHEMBL3756163 0.74 KDM4E (0.41) HPGDKEAP1RAB9ANPC1ALDH1A1
SCHEMBL3762327 0.71 KDM4E (0.38) ROCK1CDC42BPBROCK2HPGDKEAP1
SCHEMBL23850971 0.70 S100B (0.49) ROCK1CDC42BPBROCK2DHFRKEAP1
SCHEMBL4235717 0.70 CHKA (0.38) ROCK1CDC42BPBROCK2CDC42BPAHPGD
SCHEMBL15415550 0.70 CHKA (0.38) ROCK1CDC42BPBROCK2CDC42BPAHPGD
SCHEMBL14941440 0.66 GAA (0.38) ROCK1CDC42BPBROCK2CDC42BPAKEAP1
SCHEMBL21326594 0.66 ALDH1A1 (0.40) ROCK1CDC42BPBROCK2CDC42BPAKEAP1
SCHEMBL24673119 0.66 ROCK1 (1.00) ROCK1CDC42BPBROCK2CDC42BPA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103091-A1 PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF TRANSTECH PHARMA, INC. (US) 2011-08-25 WO disclosed