SCHEMBL23535339

SCHEMBL23535339

O=C1CCNC(=O)C1N1Cc2cccc(-c3ccccc3)c2C1=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 4/20 0.41
PARP11 Q9NR21 4/20 0.41
CRBN Q96SW2 3/20 0.38
PARP1 P09874 5/20 0.37
ANPEP P15144 2/20 0.36
IL1RN P18510 1/20 0.36
ERAP2 Q6P179 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
PDPK1 O15530 1/20 0.36
PRCP P42785 1/20 0.35
KMT2A Q03164 1/20 0.35
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR7 P34969 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23535409 0.82 HTR2C (0.40) CRBNPARP1KMT2AHTR2CHTR2B
SCHEMBL21997911 0.73 CRBN (0.55) CRBNPARP1HTR2CHTR2B
SCHEMBL23534354 0.73 CRBN (0.73) CRBN
SCHEMBL4345609 0.72 CRBN (0.56) PARP10PARP11CRBNPARP1HTR2C
SCHEMBL5504364 0.72 CRBN (0.39) CRBNPARP1ANPEPIL1RNERAP2
SCHEMBL29502600 0.71 CRBN (0.46) PARP10PARP11CRBNPARP1PDPK1
SCHEMBL27008204 0.71 CRBN (0.47) PARP10PARP11CRBNPARP1PDPK1
SCHEMBL29502372 0.71 CRBN (0.47) PARP10PARP11CRBNPARP1PDPK1
SCHEMBL23880787 0.68 IKZF2 (0.45)
SCHEMBL4087446 0.67 HTR3A (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021126973-A1 COMPOUNDS MODULATING PROTEIN RECRUITMENT AND/OR DEGRADATION ORIONIS BIOSCIENCES, INC. (US) 2021-06-24 WO disclosed