SCHEMBL2354840

SCHEMBL2354840

CC(O)C=CC(N)=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2354839 1.00
SCHEMBL14520488 1.00
SCHEMBL14307543 1.00
SCHEMBL20197695 1.00
SCHEMBL717707 0.80
SCHEMBL2486910 0.80 GABRP (0.40)
SCHEMBL4114676 0.80
SCHEMBL16654271 0.78
SCHEMBL5355929 0.77 GABRP (0.36)
SCHEMBL332969 0.77 ALDH1A1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3851900-B1 MONOMER COMPOSITION FOR CONTACT LENS, POLYMER THEREOF, CONTACT LENS, AND PRODUCTION METHOD THEREOF NOF CORP (JP) 2024-07-03 EP claimed
EP-3960779-B1 MONOMER COMPOSITION FOR CONTACT LENSES, POLYMER FOR CONTACT LENSES AND METHOD FOR PRODUCING SAME, AND CONTACT LENS AND METHOD FOR PRODUCING SAME NOF CORP (JP) 2024-03-13 EP claimed
EP-3578338-B1 MODEL MATERIAL INK SET, SUPPORT MATERIAL COMPOSITION, INK SET, THREE-DIMENSIONAL SHAPED OBJECT, AND METHOD FOR MANUFACTURING THREE-DIMENSIONAL SHAPED OBJECT MAXELL LTD (JP) 2023-05-10 EP claimed
EP-3689952-B1 SYRINGE GASKET SUMITOMO RUBBER IND (JP) 2022-07-20 EP claimed
EP-2894191-B1 SURFACE MODIFICATION METHOD AND SURFACE-MODIFIED ELASTIC BODY SUMITOMO RUBBER IND (JP) 2020-03-18 EP claimed
EP-3064538-B1 SURFACE MODIFICATION METHOD AND SURFACE-MODIFIED ELASTIC BODY SUMITOMO RUBBER IND (JP) 2018-09-12 EP claimed
EP-2505622-B1 Ink composition and image forming method FUJIFILM CORP (JP) 2014-01-29 EP claimed
EP-1746114-B1 WATER-SOLUBLE THICKENER AND COSMETIC PREPARATION CONTAINING SAME SHISEIDO CO LTD (JP) 2012-06-13 EP claimed
EP-0051476-B1 MODIFIED POLYURETHANE LIQUID POLYMER COMPOSITIONS AND THEIR PREPARATION OLIN CORPORATION (US) 1986-02-19 EP claimed
EP-0076126-B1 MODIFIED POLYURETHANE LIQUID POLYMER COMPOSITIONS OLIN CORPORATION (US) 1986-01-22 EP claimed
EP-3474954-B1 METHOD FOR OBTAINING A DIGLYCOSIDE-ENRICHED ARMERIA MARITIMA EXTRACT, AND USE THEREOF IN COSMETICS SOC DEXPLOITATION DE PRODUITS POUR LES INDUSTRIES CHIMIQUES SEPPIC (FR) 2023-11-29 EP disclosed
EP-3554458-B1 USE OF A HYDROCARBON MIXTURE TO IMPROVE THE SENSORIAL PROPERTIES OF GLYCERIN-BASED OIL-IN-WATER EMULSIONS SOC DEXPLOITATION DE PRODUITS POUR LES INDUSTRIES CHIMIQUES SEPPIC (FR) 2023-06-28 EP disclosed
EP-4165013-A1 METHOD FOR PREPARING AN N-ACYL AMINO ACID BY DIRECT AMIDIFICATION OF A FATTY ACID AT HIGH TEMPERATURE Société d'Exploitation de Produits pour les Industries Chimiques SEPPIC (FR) 2023-04-19 EP disclosed
EP-3773436-B1 USE OF SORBITYL POLYRHAMNOSIDES AS HUMAN SKIN LIGHTENING AGENTS SOC DEXPLOITATION DE PRODUITS POUR LES INDUSTRIES CHIMIQUES SEPPIC (FR) 2022-06-01 EP disclosed
EP-3723720-B1 NEW POLYOL POLYRHAMNOSIDES, PROCESS FOR THE PREPARATION THEREOF, AND COSMETIC AND/OR PHARMACEUTICAL COMPOSITION COMPRISING SAME SOC DEXPLOITATION DE PRODUITS POUR LES INDUSTRIES CHIMIQUES SEPPIC (FR) 2022-01-05 EP disclosed
US-20120330030-A1 Enantioselective Synthesis of y-amino-a, B-unsuturated carboxylic acid derivatives ACEMOGLU MURAT (CH) 2012-12-27 US disclosed
US-8288566-B2 Enantioselective synthesis of γ-amino-αβ-unsaturated carboxylic acid derivatives NOVARTIS AG (CH) 2012-10-16 US disclosed
US-20110263873-A1 Enantioselective Synthesis of y-amino-alpha beta-unsaturated carboxylic acid derivatives NOVARTIS AG (CH) 2011-10-27 US disclosed
EP-2358663-A1 ENANTIOSELECTIVE SYNTHESIS OF -AMINO- , -UNSATURATED CARBOXYLIC ACID DERIVATIVES Novartis AG (CH) 2011-08-24 EP disclosed
WO-2010055162-A1 ENANTIOSELECTIVE SYNTHESIS OF γ-AMINO-α,β-UNSATURATED CARBOXYLIC ACID DERIVATIVES NOVARTIS AG (CH) 2010-05-20 WO disclosed