SCHEMBL2356982

SCHEMBL2356982

Cc1ccc(Nc2cc(-n3cccc3)cc(C(F)(F)F)c2)cc1NC(=O)c1csc2c(N)ncnc12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 13/20 0.46
BRAF P15056 10/20 0.46
CSF1R P07333 10/20 0.46
DDR2 Q16832 6/20 0.46
DDR1 Q08345 5/20 0.46
ARAF P10398 1/20 0.43
KIT P10721 1/20 0.42
KDR P35968 2/20 0.41
FGFR1 P11362 1/20 0.41
TEK Q02763 1/20 0.41
MELK Q14680 1/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
EPHB2 P29323 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2359504 0.92 ABL1 (0.48) RAF1BRAFCSF1RDDR2DDR1
SCHEMBL2356986 0.90 CSF1R (0.49) RAF1BRAFCSF1RKITKDR
SCHEMBL2312566 0.82 CSF1R (0.49) RAF1BRAFCSF1RDDR2DDR1
SCHEMBL12432625 0.81 RAF1 (0.66) RAF1BRAFKITKDRPDGFRB
SCHEMBL2359009 0.81 EPHB2 (0.53) RAF1BRAFCSF1RABL1BCR
SCHEMBL12433866 0.81 CSF1R (0.53) RAF1BRAFCSF1RDDR2DDR1
SCHEMBL14717831 0.80 CSF1R (0.63) RAF1BRAFCSF1RDDR2DDR1
SCHEMBL2313222 0.80 CSF1R (0.66) RAF1BRAFCSF1RDDR2DDR1
SCHEMBL2357420 0.79 ABL1 (0.51) RAF1BRAFCSF1RABL1BCR
SCHEMBL2318397 0.79 CSF1R (0.51) RAF1BRAFCSF1RDDR2DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP claimed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO claimed
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed