SCHEMBL2359504

SCHEMBL2359504

Cc1ccc(Nc2cc(-n3ccnc3)cc(C(F)(F)F)c2)cc1NC(=O)c1csc2c(N)ncnc12

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 6/20 0.48
BCR P11274 1/20 0.48
RAF1 P04049 11/20 0.46
BRAF P15056 11/20 0.46
CSF1R P07333 5/20 0.46
DDR1 Q08345 5/20 0.46
DDR2 Q16832 5/20 0.46
SRC P12931 1/20 0.42
EPHB2 P29323 1/20 0.42
ARAF P10398 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2356982 0.92 RAF1 (0.46) ABL1BCRRAF1BRAFCSF1R
SCHEMBL2312566 0.91 CSF1R (0.49) ABL1BCRRAF1BRAFCSF1R
SCHEMBL2356986 0.82 CSF1R (0.49) RAF1BRAFCSF1RSRC
SCHEMBL2359009 0.81 EPHB2 (0.53) ABL1BCRRAF1BRAFCSF1R
SCHEMBL12432625 0.81 RAF1 (0.66) ABL1BCRRAF1BRAFSRC
SCHEMBL14717831 0.80 CSF1R (0.63) RAF1BRAFCSF1RDDR1DDR2
SCHEMBL2357420 0.79 ABL1 (0.51) ABL1BCRRAF1BRAFCSF1R
SCHEMBL12433866 0.79 CSF1R (0.53) RAF1BRAFCSF1RDDR1DDR2
SCHEMBL12433888 0.79 ABL1 (0.57) ABL1BCRRAF1BRAFCSF1R
SCHEMBL2318397 0.77 CSF1R (0.51) ABL1RAF1BRAFCSF1RDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed