SCHEMBL2359009

SCHEMBL2359009

CNc1ncnc2c(C(=O)Nc3cc(Nc4cc(-n5cnc(C)c5)cc(C(F)(F)F)c4)ccc3C)csc12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHB2 P29323 1/20 0.53
RAF1 P04049 1/20 0.50
BRAF P15056 3/20 0.49
HCK P08631 1/20 0.49
NR2C2 P49116 1/20 0.49
BTK Q06187 1/20 0.49
CSF1R P07333 1/20 0.49
MAP4K2 Q12851 1/20 0.49
ABL1 P00519 5/20 0.48
BCR P11274 3/20 0.48
NR2E1 Q9Y466 4/20 0.47
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2357420 0.92 ABL1 (0.51) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL12433483 0.91 CSF1R (0.62) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL2359059 0.89 EPHB2 (0.50) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL2359007 0.89 CSF1R (0.47) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL2358403 0.88 BRAF (0.52) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL14110085 0.85 ABL1 (0.56) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL14717948 0.84 CSF1R (0.59) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL14717868 0.83 CSF1R (0.59) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL12433883 0.83 CSF1R (0.59) EPHB2RAF1BRAFHCKNR2C2
SCHEMBL12432625 0.83 RAF1 (0.66) EPHB2RAF1BRAFHCKNR2C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed