SCHEMBL2358009

SCHEMBL2358009

OCN1Cc2ccccc2C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.46
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
NOTUM Q6P988 1/20 0.43
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
PHGDH O43175 1/20 0.39
MGLL Q99685 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14067117 0.84 HDAC3 (0.54) CARM1ALDH1A1MEN1KMT2AHDAC3
SCHEMBL29367146 0.80 ALDH1A1 (0.52) CARM1ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL377728 0.80 ALDH1A1 (0.52) CARM1ALDH1A1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL25366946 0.78 ALDH1A1 (0.50) CARM1ALDH1A1CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL30528641 0.78 ALDH1A1 (0.50) CARM1ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL30072993 0.78 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP2D6CYP2C19ADRA1D
SCHEMBL9378373 0.77 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2D6CYP2C19HDAC3
SCHEMBL14067241 0.77 PDK2 (0.46)
SCHEMBL22295970 0.76 ALDH1A1 (0.47) CARM1ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL14067201 0.75 DPP8 (0.43) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3651768-A1 HETEROCYCLIC INHIBITORS OF ATR KINASE Board of Regents, The University of Texas System (US) 2020-05-20 EP disclosed
WO-2019014618-A1 HETEROCYCLIC INHIBITORS OF ATR KINASE BOARD OF REGENTS, UNIVERSITY OF TEXAS SYSTEM (US) 2019-01-17 WO disclosed
WO-2011091410-A1 TRPV4 ANTAGONISTS GLAXOS SMITHKLINE LLC (US) 2011-07-28 WO disclosed