SCHEMBL2358403

SCHEMBL2358403

Cc1cn(-c2cc(Nc3ccc(C)c(NC(=O)c4csc5c(NC6CCN(C)CC6)ncnc45)c3)cc(C(F)(F)F)c2)cn1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.52
ABL1 P00519 6/20 0.51
SRC P12931 2/20 0.51
BCR P11274 3/20 0.49
EPHB2 P29323 1/20 0.47
RAF1 P04049 1/20 0.45
CSF1R P07333 3/20 0.45
HCK P08631 1/20 0.45
NR2C2 P49116 1/20 0.45
BTK Q06187 1/20 0.45
DDR1 Q08345 2/20 0.44
DDR2 Q16832 2/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44
NTRK1 P04629 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14717773 0.92 CSF1R (0.55) BRAFABL1SRCBCREPHB2
SCHEMBL2358401 0.90 BRAF (0.46) BRAFABL1SRCBCREPHB2
SCHEMBL14110085 0.90 ABL1 (0.56) BRAFABL1SRCBCREPHB2
SCHEMBL2359009 0.88 EPHB2 (0.53) BRAFABL1BCREPHB2RAF1
SCHEMBL12433475 0.88 ABL1 (0.63) BRAFABL1SRCBCREPHB2
SCHEMBL12432449 0.87 CSF1R (0.58) BRAFABL1SRCBCREPHB2
SCHEMBL2357420 0.86 ABL1 (0.51) BRAFABL1BCREPHB2RAF1
SCHEMBL12433869 0.86 CSF1R (0.57) BRAFABL1SRCBCREPHB2
SCHEMBL14716921 0.84 CSF1R (0.63) BRAFABL1SRCRAF1CSF1R
SCHEMBL2359059 0.84 EPHB2 (0.50) BRAFABL1BCREPHB2RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP claimed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO claimed
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed