SCHEMBL23587349

SCHEMBL23587349

COC(O)c1nn(C(F)F)c2cc(O)ccc12

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.35
HTR3A P46098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19127270 0.75 ELANE (0.42) HTR3A
SCHEMBL30711997 0.75 ELANE (0.42) HTR3A
SCHEMBL15723742 0.66 GRM4 (0.43) ESR1
SCHEMBL27702080 0.62 ABL1 (0.41) ESR1
SCHEMBL492329 0.61 ALDH1A1 (0.44) HTR3A
SCHEMBL30147561 0.61 CSNK2A1 (0.42)
SCHEMBL19128146 0.61 ELANE (0.42)
SCHEMBL29301466 0.61 CSNK2A1 (0.42)
SCHEMBL31632866 0.60 NOTUM (0.42)
SCHEMBL23093693 0.60 ELANE (0.49) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3652168-B1 5-MEMBERED AND BICYCLIC HETEROCYCLIC AMIDES AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2021-06-30 EP disclosed