SCHEMBL30711997

SCHEMBL30711997

COC(=O)c1nn(C(F)F)c2cc(O)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 9/20 0.42
PLAU P00749 5/20 0.42
F2 P00734 4/20 0.42
HTR3A P46098 1/20 0.41
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA14 Q9ULX7 3/20 0.39
PDK2 Q15119 1/20 0.39
PDK4 Q16654 1/20 0.39
CTRB1 P17538 2/20 0.38
MAPT P10636 4/20 0.37
KDM4E B2RXH2 3/20 0.37
PKM P14618 3/20 0.37
HPGD P15428 2/20 0.37
ALOX15 P16050 2/20 0.37
HSD17B10 Q99714 2/20 0.37
GAA P10253 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19127270 1.00 ELANE (0.42) ELANEPLAUF2HTR3ACA12
SCHEMBL19128146 0.86 ELANE (0.42) ELANEPLAUF2CTRB1KDM4E
SCHEMBL19127362 0.85 ELANE (0.50) ELANEPLAUF2CTRB1MAPT
SCHEMBL23093693 0.85 ELANE (0.49) ELANEPLAUF2HTR3AMAPT
SCHEMBL23093689 0.85 ELANE (0.41) ELANEPLAUF2CTRB1MAPT
SCHEMBL28568174 0.82 ELANE (0.58) ELANEPLAUF2HTR3AMAPT
SCHEMBL30711990 0.79 HTR3A (0.51) ELANEPLAUF2HTR3AKDM4E
SCHEMBL19127310 0.79 HTR3A (0.51) ELANEPLAUF2HTR3AKDM4E
SCHEMBL23093692 0.78 ELANE (0.43) ELANEPLAUF2HTR3ACTRB1
SCHEMBL19149244 0.78 ROCK2 (0.53) ELANEPLAUF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110869363-B 5-membered and bicyclic heterocyclic amides as ROCK inhibitors 百时美施贵宝公司 2024-01-05 CN disclosed