SCHEMBL23587447

SCHEMBL23587447

C=C(CN)Cc1ccc(CC(C)c2ccc(C)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.49
ESR2 Q92731 2/20 0.49
ACHE P22303 1/20 0.37
HPGD P15428 1/20 0.36
STAT3 P40763 1/20 0.35
CNR2 P34972 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
EPHX1 P07099 1/20 0.34
CNR1 P21554 1/20 0.33
HCRTR2 O43614 2/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
PSMB8 P28062 1/20 0.33
PSMB5 P28074 1/20 0.33
AKR1C3 P42330 1/20 0.32
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547203 0.80 ESR1 (0.65) ESR1ESR2ACHESTAT3CYP1A2
SCHEMBL1954002 0.75 ESR1 (0.85) ESR1ESR2ACHEHPGDCYP1A2
SCHEMBL21699675 0.75 ESR1 (0.55) ESR1ESR2ACHESTAT3CYP1A2
SCHEMBL1841040 0.75 ESR1 (0.85) ESR1ESR2ACHEHPGDCYP1A2
SCHEMBL6546854 0.73 ESR1 (0.57) ESR1ESR2ACHESTAT3HCRTR2
SCHEMBL6546983 0.73 ESR1 (0.57) ESR1ESR2ACHESTAT3HCRTR2
SCHEMBL2844467 0.72 ESR1 (0.55) ESR1ESR2ACHECNR2
SCHEMBL2844291 0.71 ESR1 (0.53) ESR1ESR2CYP2A6TAAR1HCRTR2
SCHEMBL5313594 0.71 ESR1 (0.53) ESR1ESR2ACHECNR2CYP2A6
SCHEMBL15070045 0.70 ESR1 (0.53) ESR1ESR2ACHESTAT3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3509583-B1 ESTROGEN RECEPTOR LIGANDS, COMPOSITIONS AND METHODS RELATED THERETO UNIV CALIFORNIA (US) 2021-06-30 EP disclosed